LY339434 [Ligand Id: 4246] activity data from GtoPdb

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  • GluK1 in Human [GtoPdb: 450] [UniProtKB: P39086]
  • This target only has 1 pki data point
  • 7.89
1 _lig_chart_1 GluK1 Human
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  • GluK2 in Human [GtoPdb: 451] [UniProtKB: Q13002]
  • This target only has 1 pki data point
  • 4.92
2 _lig_chart_2 GluK2 Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
GluK1 in Human [GtoPdb: 450] [UniProtKB: P39086]
GtoPdb - - 7.89 pKi 13 nM Ki Neuropharmacology (1998) 37: 1261-7 [PMID:9849663]
GluK2 in Human [GtoPdb: 451] [UniProtKB: Q13002]
GtoPdb - - 4.92 pKi 12040 nM Ki Neuropharmacology (1998) 37: 1261-7 [PMID:9849663]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.