ChEMBL ligand: CHEMBL211502 (Phenamil)
ENaC α/Amiloride-sensitive sodium channel alpha-subunit in Human [ChEMBL: CHEMBL1791] [GtoPdb: 738] [UniProtKB: P37088] This target only has 0 pki data point 1 CHEMBL211502_lig_chart_1 Amiloride-sensitive sodium channel alpha-subunit Human There should be some charts here, you may need to enable JavaScript!
TRPP2 in Human [GtoPdb: 505] [UniProtKB: Q9P0L9] This target only has 0 pki data point 2 CHEMBL211502_lig_chart_2 TRPP2 Human There should be some charts here, you may need to enable JavaScript!

DB	Assay description	Assay Type	Standard value	Standard parameter	Original value	Original units	Original parameter	Reference
ENaC α/Amiloride-sensitive sodium channel alpha-subunit in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL1791] [GtoPdb: 738] [UniProtKB: P37088]
ChEMBL	Inhibition of dog bronchi prototypical epithelial sodium channel by electrophysiological assay	B	6.4	pIC50	401	nM	IC50	J. Med. Chem. (2006) 49: 4098-4115 [PMID:16821771]
TRPP2 in Human [GtoPdb: 505] [UniProtKB: Q9P0L9]
GtoPdb	-	-	6.9	pIC50	140	nM	IC50

ChEMBL data shown on this page come from version 27:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]