bromocresol green [Ligand Id: 4530] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL145704 (Bromocresol Green)
  • OATP2A1/Solute carrier organic anion transporter family member 2A1 in Rat [ChEMBL: CHEMBL2073680] [GtoPdb: 1223] [UniProtKB: Q00910]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
OATP2A1/Solute carrier organic anion transporter family member 2A1 in Rat (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL2073680] [GtoPdb: 1223] [UniProtKB: Q00910]
GtoPdb - - 5.44 pKi 3600 nM Ki Science (1995) 268: 866-9 [PMID:7754369]
ChEMBL TP_TRANSPORTER: inhibition of PGF2alpha uptake in PGT-expressing HeLa cells F 5.44 pKi 3600 nM Ki Science (1995) 268: 866-869 [PMID:7754369]

ChEMBL data shown on this page come from version 28:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]