[3H]ZM 241385 [Ligand Id: 455] activity data from GtoPdb and ChEMBL
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| ChEMBL ligand: CHEMBL1628684 (ZM-241385) |
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| A2A receptor in Human [GtoPdb: 19] [UniProtKB: P29274] | ||||||||
| GtoPdb | - | - | 9.1 | pKd | 0.8 | nM | Kd |
Eur J Pharmacol (2001) 411: 205-10 [PMID:11164377]; Biochem Pharmacol (2000) 60: 661-8 [PMID:10927024] |
| A2B receptor in Human [GtoPdb: 20] [UniProtKB: P29275] | ||||||||
| GtoPdb | - | - | 7.9 | pKd | - | - | - |
Biochem Pharmacol (2001) 62: 1163-73 [PMID:11705449]; Biochem Pharmacol (2004) 68: 305-12 [PMID:15194002]; Drug Des Discov (1999) 16: 217-26 [PMID:10624567] |
ChEMBL data shown on this page come from version 33:
Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]
