[125I]BE-2254 [Ligand Id: 500] activity data from GtoPdb

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  • α1A-adrenoceptor in Human [GtoPdb: 22] [UniProtKB: P35348]
  • This target only has 0 pki data point
  • 0
1 _lig_chart_1 α1A-adrenoceptor Human
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  • α1B-adrenoceptor in Human [GtoPdb: 23] [UniProtKB: P35368]
  • This target only has 0 pki data point
  • 0
2 _lig_chart_2 α1B-adrenoceptor Human
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  • α1D-adrenoceptor in Human [GtoPdb: 24] [UniProtKB: P25100]
  • This target only has 0 pki data point
  • 0
3 _lig_chart_3 α1D-adrenoceptor Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
α1A-adrenoceptor in Human [GtoPdb: 22] [UniProtKB: P35348]
GtoPdb - - 9.9 pKd - - - Pharmacol Ther (2000) 88: 281-309 [PMID:11337028];
J Pharmacol Exp Ther (1995) 272: 134-42 [PMID:7815325]
α1B-adrenoceptor in Human [GtoPdb: 23] [UniProtKB: P35368]
GtoPdb - - 9.9 pKd - - - Pharmacol Ther (2000) 88: 281-309 [PMID:11337028];
J Pharmacol Exp Ther (1995) 272: 134-42 [PMID:7815325]
α1D-adrenoceptor in Human [GtoPdb: 24] [UniProtKB: P25100]
GtoPdb - - 9.9 pKd - - - J Pharmacol Exp Ther (1995) 272: 134-42 [PMID:7815325]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.