EHNA [Ligand Id: 5179] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL1257094
  • Adenosine deaminase in Human [GtoPdb: 1230] [UniProtKB: P00813]
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  • phosphodiesterase 2A in Human [GtoPdb: 1297] [UniProtKB: O00408]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Adenosine deaminase in Human [GtoPdb: 1230] [UniProtKB: P00813]
GtoPdb - - 8.8 pKi - - - Biochem. Pharmacol. (1977) 26: 359-67 [PMID:849330]
phosphodiesterase 2A in Human [GtoPdb: 1297] [UniProtKB: O00408]
GtoPdb - - 5.3 pIC50 5010 nM IC50 Cell. Signal. (1996) 8: 97-110 [PMID:8730511]

ChEMBL data shown on this page come from version 26:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]