galanin(2-11) [Ligand Id: 5357] activity data from GtoPdb

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  • GAL1 receptor in Human [GtoPdb: 243] [UniProtKB: P47211]
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  • GAL2 receptor in Human [GtoPdb: 244] [UniProtKB: O43603]
  • GAL2 receptor in Rat [GtoPdb: 244] [UniProtKB: O08726]
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  • GAL3 receptor in Human [GtoPdb: 245] [UniProtKB: O60755]
  • GAL3 receptor in Rat [GtoPdb: 245] [UniProtKB: O88626]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
GAL1 receptor in Human [GtoPdb: 243] [UniProtKB: P47211]
GtoPdb - - 5.3 pKi >5000 nM Ki Neuropeptides (2005) 39: 143-6 [PMID:15944002]
GtoPdb - - 6.06 pIC50 879 nM IC50 Proc Natl Acad Sci USA (2001) 98: 9960-4 [PMID:11481429]
GAL2 receptor in Human [GtoPdb: 244] [UniProtKB: O43603]
GtoPdb - - 7.78 pKi 16.6 nM Ki Neuropeptides (2009) 43: 187-92 [PMID:19467704]
GAL2 receptor in Rat [GtoPdb: 244] [UniProtKB: O08726]
GtoPdb - - 7.06 pKi 88 nM Ki Neuropeptides (2005) 39: 165-7 [PMID:15944007]
GtoPdb - - 8.75 pIC50 1.76 nM IC50 Proc Natl Acad Sci USA (2001) 98: 9960-4 [PMID:11481429]
GAL3 receptor in Human [GtoPdb: 245] [UniProtKB: O60755]
GtoPdb - - 6.7 pKi 199 nM Ki Neuropeptides (2009) 43: 187-92 [PMID:19467704]
GAL3 receptor in Rat [GtoPdb: 245] [UniProtKB: O88626]
GtoPdb - - 6.57 pKi 271 nM Ki Neuropeptides (2005) 39: 165-7 [PMID:15944007]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.