GS9667 [Ligand Id: 5593] activity data from GtoPdb

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  • A1 receptor in Human [GtoPdb: 18] [UniProtKB: P30542]
  • This target only has 1 pki data point
1 _lig_chart_1 A1 receptor Human
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  • A2A receptor in Human [GtoPdb: 19] [UniProtKB: P29274]
  • This target only has 1 pki data point
2 _lig_chart_2 A2A receptor Human
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  • A2B receptor in Human [GtoPdb: 20] [UniProtKB: P29275]
  • This target only has 1 pki data point
3 _lig_chart_3 A2B receptor Human
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  • A3 receptor in Human [GtoPdb: 21] [UniProtKB: P0DMS8]
  • This target only has 1 pki data point
4 _lig_chart_4 A3 receptor Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
A1 receptor in Human [GtoPdb: 18] [UniProtKB: P30542]
GtoPdb - - 7.26 pKi 55 nM Ki Expert Opin Investig Drugs (2008) 17: 1901-10 [PMID:19012505]
A2A receptor in Human [GtoPdb: 19] [UniProtKB: P29274]
GtoPdb - - 5 pKi >10000 nM Ki Expert Opin Investig Drugs (2008) 17: 1901-10 [PMID:19012505]
A2B receptor in Human [GtoPdb: 20] [UniProtKB: P29275]
GtoPdb - - 4.3 pKi >50000 nM Ki Expert Opin Investig Drugs (2008) 17: 1901-10 [PMID:19012505]
A3 receptor in Human [GtoPdb: 21] [UniProtKB: P0DMS8]
GtoPdb - - 6 pKi >1000 nM Ki Expert Opin Investig Drugs (2008) 17: 1901-10 [PMID:19012505]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.