β2-adrenoceptor in Human [GtoPdb: 29] [UniProtKB: P07550] 4.3 1 _lig_chart_1 β2-adrenoceptor Human There should be some charts here, you may need to enable JavaScript!
GPR83 in Mouse [GtoPdb: 119] [UniProtKB: P30731] This target only has 0 pki data point 0 2 _lig_chart_2 GPR83 Mouse There should be some charts here, you may need to enable JavaScript!
glycine receptor α1 subunit in Human [GtoPdb: 423] [UniProtKB: P23415] This target only has 0 pki data point 0 3 _lig_chart_3 glycine receptor α1 subunit Human There should be some charts here, you may need to enable JavaScript!
glycine receptor α2 subunit in Human [GtoPdb: 424] [UniProtKB: P23416] This target only has 0 pki data point 0 4 _lig_chart_4 glycine receptor α2 subunit Human There should be some charts here, you may need to enable JavaScript!
glycine receptor α3 subunit in Human [GtoPdb: 425] [UniProtKB: O75311] This target only has 0 pki data point 0 5 _lig_chart_5 glycine receptor α3 subunit Human There should be some charts here, you may need to enable JavaScript!
glycine receptor β subunit in Human [GtoPdb: 427] [UniProtKB: P48167] This target only has 0 pki data point 0 6 _lig_chart_6 glycine receptor β subunit Human There should be some charts here, you may need to enable JavaScript!
TRPA1 in Mouse [GtoPdb: 485] [UniProtKB: Q8BLA8] This target only has 0 pki data point 0 7 _lig_chart_7 TRPA1 Mouse There should be some charts here, you may need to enable JavaScript!
TRPM1 in Human [GtoPdb: 493] [UniProtKB: Q7Z4N2] This target only has 0 pki data point 0 8 _lig_chart_8 TRPM1 Human There should be some charts here, you may need to enable JavaScript!
TRPM2 in Human [GtoPdb: 494] [UniProtKB: O94759] This target only has 0 pki data point 0 9 _lig_chart_9 TRPM2 Human There should be some charts here, you may need to enable JavaScript!
ZAC in Human [GtoPdb: 587] [UniProtKB: Q401N2] This target only has 0 pki data point 0 10 _lig_chart_10 ZAC Human There should be some charts here, you may need to enable JavaScript!
ASIC1 in Human [GtoPdb: 684] [UniProtKB: P78348] This target only has 0 pki data point 0 11 _lig_chart_11 ASIC1 Human There should be some charts here, you may need to enable JavaScript!
ASIC3 in Human [GtoPdb: 686] [UniProtKB: Q9UHC3] This target only has 0 pki data point 0 12 _lig_chart_12 ASIC3 Human There should be some charts here, you may need to enable JavaScript!
ClC-4 in Human [GtoPdb: 703] [UniProtKB: P51793] This target only has 0 pki data point 0 13 _lig_chart_13 ClC-4 Human There should be some charts here, you may need to enable JavaScript!
Maxi Cl- in Human [GtoPdb: 709] This target only has 0 pki data point 0 14 _lig_chart_14 Maxi Cl- Human There should be some charts here, you may need to enable JavaScript!
Hv1 in Human [GtoPdb: 746] [UniProtKB: Q96D96] This target only has 0 pki data point 0 15 _lig_chart_15 Hv1 Human There should be some charts here, you may need to enable JavaScript!

DB	Assay description	Assay Type	Standard value	Standard parameter	Original value	Original units	Original parameter	Reference
β2-adrenoceptor in Human [GtoPdb: 29] [UniProtKB: P07550]
GtoPdb	-	-	3.3	pKi	-	-	-	J Biol Chem (2003) 278: 352-6 [PMID:12409304]; Mol Pharmacol (2002) 61: 65-72 [PMID:11752207]
GtoPdb	-	-	5.3	pKi	-	-	-	J Biol Chem (2003) 278: 352-6 [PMID:12409304]; Mol Pharmacol (2002) 61: 65-72 [PMID:11752207]
GPR83 in Mouse [GtoPdb: 119] [UniProtKB: P30731]
GtoPdb	-	-	5	pEC50	10200	nM	EC50	PLoS ONE (2013) 8: e53347 [PMID:23335960]
glycine receptor α1 subunit in Human [GtoPdb: 423] [UniProtKB: P23415]
GtoPdb	-	-	4.8	pIC50	15000	nM	IC50
GtoPdb	-	-	7.4	pEC50	37	nM	EC50
glycine receptor α2 subunit in Human [GtoPdb: 424] [UniProtKB: P23416]
GtoPdb	-	-	3.4	pIC50	360000	nM	IC50
GtoPdb	-	-	6.3	pEC50	540	nM	EC50
glycine receptor α3 subunit in Human [GtoPdb: 425] [UniProtKB: O75311]
GtoPdb	-	-	3.8	pIC50	150000	nM	IC50
glycine receptor β subunit in Human [GtoPdb: 427] [UniProtKB: P48167]
GtoPdb	-	-	3.7	pIC50	180000	nM	IC50
GtoPdb	-	-	4.9	pIC50	13000	nM	IC50
TRPA1 in Mouse [GtoPdb: 485] [UniProtKB: Q8BLA8]
GtoPdb	Calcium imaging	-	2.3	pEC50	-	-	-	Nat Chem Biol (2009) 5: 183-90 [PMID:19202543]; Proc Natl Acad Sci USA (2009) 106: 8374-9 [PMID:19416844]
TRPM1 in Human [GtoPdb: 493] [UniProtKB: Q7Z4N2]
GtoPdb	-	-	6	pIC50	1000	nM	IC50
TRPM2 in Human [GtoPdb: 494] [UniProtKB: O94759]
GtoPdb	-	-	6	pIC50	1000	nM	IC50
ZAC in Human [GtoPdb: 587] [UniProtKB: Q401N2]
GtoPdb	-	-	3.7	pEC50	-	-	EC50	J Biol Chem (2003) 278: 712-7 [PMID:12381728]; Biochem Pharmacol (2016) 103: 109-17 [PMID:26872532]
ASIC1 in Human [GtoPdb: 684] [UniProtKB: P78348]
GtoPdb	-	-	8.2	pIC50	~7	nM	IC50	J Neurosci (2004) 24: 8678-89 [PMID:15470133]
ASIC3 in Human [GtoPdb: 686] [UniProtKB: Q9UHC3]
GtoPdb	-	-	4.2	pIC50	61000	nM	IC50	Neuroscience (2010) 169: 574-83 [PMID:20580786]
ClC-4 in Human [GtoPdb: 703] [UniProtKB: P51793]
GtoPdb	-	-	4.3	pIC50	50000	nM	IC50	Biophys J (2008) 95: 4668-75 [PMID:18658230]
Maxi Cl- in Human [GtoPdb: 709]
GtoPdb	-	-	4.3	pIC50	50000	nM	IC50	Biophys J (2008) 95: 4668-75 [PMID:18658230]
Hv1 in Human [GtoPdb: 746] [UniProtKB: Q96D96]
GtoPdb	-	-	6.3	pIC50	~500	nM	IC50