YSFKPMPLaR [Ligand Id: 5776] activity data from GtoPdb

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  • C3a receptor in Human [GtoPdb: 31] [UniProtKB: Q16581]
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  • C5a1 receptor in Human [GtoPdb: 32] [UniProtKB: P21730]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
C3a receptor in Human [GtoPdb: 31] [UniProtKB: Q16581]
GtoPdb - - 6.7 pEC50 220 nM EC50 J Med Chem (2010) 53: 4938-48 [PMID:20527893]
C5a1 receptor in Human [GtoPdb: 32] [UniProtKB: P21730]
GtoPdb - - 6.7 pIC50 200 nM IC50 J Med Chem (1997) 40: 877-84 [PMID:9083476]
GtoPdb - - 5.5 pEC50 3240 nM EC50 Inflammation (2001) 25: 171-7 [PMID:11403208]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.