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ChEMBL ligand: CHEMBL3286797 (Pf-04418948) |
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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BLT1 receptor/Leukotriene B4 receptor 1 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3911] [GtoPdb: 267] [UniProtKB: Q15722] | ||||||||
ChEMBL | LTB4 (h) (BLT1) CEREP ligand profiling | B | 5.32 | pKi | 4800 | nM | Ki | Data for DCP probe PF-04418948 |
ChEMBL | LTB4 (h) (BLT1) CEREP ligand profiling | B | 5.01 | pIC50 | 9700 | nM | IC50 | Data for DCP probe PF-04418948 |
EP2 receptor/Prostanoid EP2 receptor in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL1881] [GtoPdb: 341] [UniProtKB: P43116] | ||||||||
ChEMBL | Inhibition of binding to PTGER2 | B | 8.3 | pIC50 | 5 | nM | IC50 | Data for DCP probe PF-04418948 |
EP2 receptor in Mouse [GtoPdb: 341] [UniProtKB: Q62053] | ||||||||
Quinone reductase 2 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3959] [UniProtKB: P16083] | ||||||||
ChEMBL | ML2 (MT3) CEREP ligand profiling | B | 6.28 | pKi | 520 | nM | Ki | Data for DCP probe PF-04418948 |
ChEMBL | ML2 (MT3) CEREP ligand profiling | B | 6.28 | pIC50 | 530 | nM | IC50 | Data for DCP probe PF-04418948 |
ChEMBL data shown on this page come from version 33:
Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]