PD123177 [Ligand Id: 596] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL1188080
  • AT2 receptor in Rat [GtoPdb: 35] [UniProtKB: P35351]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
AT2 receptor in Rat [GtoPdb: 35] [UniProtKB: P35351]
GtoPdb - - 9.49 pIC50 0.32 nM IC50 Biochem Biophys Res Commun (1989) 165: 196-203 [PMID:2590220];
Regul Pept (1993) 44: 199-206 [PMID:8469774];
Mol Pharmacol (1990) 37: 347-51 [PMID:2314387]

ChEMBL data shown on this page come from version 28:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]