galmic [Ligand Id: 6119] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL1187471 (Galmic)
  • GAL1 receptor/Galanin receptor 1 in Human [ChEMBL: CHEMBL4894] [GtoPdb: 243] [UniProtKB: P47211]
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  • GAL2 receptor/Galanin receptor 2 in Rat [ChEMBL: CHEMBL5577] [GtoPdb: 244] [UniProtKB: O08726]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
GAL1 receptor/Galanin receptor 1 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL4894] [GtoPdb: 243] [UniProtKB: P47211]
ChEMBL Binding affinity to human GalR1 B 4.47 pKi 34200 nM Ki J. Med. Chem. (2010) 53: 1871-1875 [PMID:20121116]
GtoPdb - - 4.47 pKi 34200 nM Ki Neuropeptides (2005) 39: 161-3 [PMID:15944006];
Proc Natl Acad Sci USA (2004) 101: 10470-5 [PMID:15240875]
GAL2 receptor/Galanin receptor 2 in Rat (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL5577] [GtoPdb: 244] [UniProtKB: O08726]
GtoPdb - - 5 pKd >10000 nM Kd Proc Natl Acad Sci USA (2004) 101: 10470-5 [PMID:15240875];
Neuropeptides (2005) 39: 143-6 [PMID:15944002]
ChEMBL Binding affinity to rat GalR2 B 4 pKi >100000 nM Ki J. Med. Chem. (2010) 53: 1871-1875 [PMID:20121116]

ChEMBL data shown on this page come from version 28:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]