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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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BB1 receptor in Human [GtoPdb: 38] [UniProtKB: P28336] | ||||||||
GtoPdb | - | - | 8.83 | pIC50 | 1.48 | nM | IC50 | Peptides (2011) 32: 1685-99 [PMID:21729729] |
BB1 receptor in Rat [GtoPdb: 38] [UniProtKB: P24053] | ||||||||
GtoPdb | - | - | 7.89 | pKi | 13 | nM | Ki |
J Biol Chem (1997) 272: 26062-71 [PMID:9325344]; Biochemistry (1999) 38: 7307-20 [PMID:10353842] |
BB2 receptor in Human [GtoPdb: 39] [UniProtKB: P30550] | ||||||||
GtoPdb | - | - | 8.65 | pIC50 | 2.24 | nM | IC50 | Peptides (2011) 32: 1685-99 [PMID:21729729] |
BB2 receptor in Rat [GtoPdb: 39] [UniProtKB: P52500] | ||||||||
GtoPdb | - | - | 8.7 | pKi | 2 | nM | Ki |
J Biol Chem (1997) 272: 26062-71 [PMID:9325344]; Biochemistry (1999) 38: 7307-20 [PMID:10353842] |
GtoPdb | - | - | 8.97 | pIC50 | 1.08 | nM | IC50 | Peptides (2011) 32: 1685-99 [PMID:21729729] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.