[D-Phe6,β-Ala11,Phe13,Nle14]bombesin-(6-14) [Ligand Id: 632] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| BB1 receptor in Human [GtoPdb: 38] [UniProtKB: P28336] | ||||||||
| GtoPdb | - | - | 9.7 | pKi | - | - | - |
J Pharmacol Exp Ther (1999) 290: 1202-11 [PMID:10454496]; Peptides (2011) 32: 1685-99 [PMID:21729729] |
| GtoPdb | - | - | 9.68 | pIC50 | 0.21 | nM | IC50 | Peptides (2011) 32: 1685-99 [PMID:21729729] |
| BB2 receptor in Human [GtoPdb: 39] [UniProtKB: P30550] | ||||||||
| GtoPdb | - | - | 8 | pKi | 10 | nM | Ki |
J Pharmacol Exp Ther (1999) 290: 1202-11 [PMID:10454496]; J Pept Sci (2019) 25: e3224 [PMID:31743956] |
| GtoPdb | - | - | 10.32 | pIC50 | 0.05 | nM | IC50 | Peptides (2011) 32: 1685-99 [PMID:21729729] |
| BB3 receptor in Human [GtoPdb: 40] [UniProtKB: P32247] | ||||||||
| GtoPdb | - | - | 8.38 | pKi | 4.2 | nM | Ki | J Biol Chem (1997) 272: 26062-71 [PMID:9325344] |
| BB3 receptor in Mouse [GtoPdb: 40] [UniProtKB: O54798] | ||||||||
| GtoPdb | - | - | 8.82 | pKi | 1.5 | nM | Ki | J Pharmacol Exp Ther (1999) 290: 1202-11 [PMID:10454496] |
| BB3 receptor in Rat [GtoPdb: 40] [UniProtKB: Q8K418] | ||||||||
| GtoPdb | - | - | 9 | pKi | 1 | nM | Ki | J Pharmacol Exp Ther (1999) 290: 1202-11 [PMID:10454496] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
