[D-Phe6,β-Ala11,Phe13,Nle14]bombesin-(6-14) [Ligand Id: 632] activity data from GtoPdb

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  • BB1 receptor in Human [GtoPdb: 38] [UniProtKB: P28336]
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  • BB2 receptor in Human [GtoPdb: 39] [UniProtKB: P30550]
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  • BB3 receptor in Human [GtoPdb: 40] [UniProtKB: P32247]
  • BB3 receptor in Mouse [GtoPdb: 40] [UniProtKB: O54798]
  • BB3 receptor in Rat [GtoPdb: 40] [UniProtKB: Q8K418]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
BB1 receptor in Human [GtoPdb: 38] [UniProtKB: P28336]
GtoPdb - - 9.7 pKi - - - J. Pharmacol. Exp. Ther. (1999) 290: 1202-11 [PMID:10454496];
Peptides (2011) 32: 1685-99 [PMID:21729729]
GtoPdb - - 9.68 pIC50 0.21 nM IC50 Peptides (2011) 32: 1685-99 [PMID:21729729]
BB2 receptor in Human [GtoPdb: 39] [UniProtKB: P30550]
GtoPdb - - 8 pKi 10 nM Ki J. Pharmacol. Exp. Ther. (1999) 290: 1202-11 [PMID:10454496]
GtoPdb - - 10.32 pIC50 0.05 nM IC50 Peptides (2011) 32: 1685-99 [PMID:21729729]
BB3 receptor in Human [GtoPdb: 40] [UniProtKB: P32247]
GtoPdb - - 8.38 pKi 4.2 nM Ki J. Biol. Chem. (1997) 272: 26062-71 [PMID:9325344]
BB3 receptor in Mouse [GtoPdb: 40] [UniProtKB: O54798]
GtoPdb - - 8.82 pKi 1.5 nM Ki J. Pharmacol. Exp. Ther. (1999) 290: 1202-11 [PMID:10454496]
BB3 receptor in Rat [GtoPdb: 40] [UniProtKB: Q8K418]
GtoPdb - - 9 pKi 1 nM Ki J. Pharmacol. Exp. Ther. (1999) 290: 1202-11 [PMID:10454496]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.