Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
ChEMBL ligand: CHEMBL1335656 |
---|
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
There should be some charts here, you may need to enable JavaScript!
|
DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
---|---|---|---|---|---|---|---|---|
carbonic anhydrase 1 in Human [GtoPdb: 2597] [UniProtKB: P00915] | ||||||||
GtoPdb | - | - | 7.48 | pKi | 33 | nM | Ki |
Bioorg. Med. Chem. Lett. (2005) 15: 3828-33 [PMID:16039848]; Bioorg. Med. Chem. Lett. (2005) 15: 963-9 [PMID:15686894] |
carbonic anhydrase 14 in Human [GtoPdb: 2598] [UniProtKB: Q9ULX7] | ||||||||
GtoPdb | - | - | 7.57 | pKi | 27 | nM | Ki | Bioorg. Med. Chem. Lett. (2005) 15: 3828-33 [PMID:16039848] |
carbonic anhydrase 4 in Human [GtoPdb: 2599] [UniProtKB: P22748] | ||||||||
GtoPdb | - | - | 7.62 | pKi | 24 | nM | Ki | Bioorg. Med. Chem. Lett. (2005) 15: 3828-33 [PMID:16039848] |
carbonic anhydrase 12 in Human [GtoPdb: 2747] [UniProtKB: O43570] | ||||||||
GtoPdb | - | - | 8.47 | pKi | 3.4 | nM | Ki | Bioorg. Med. Chem. Lett. (2005) 15: 963-9 [PMID:15686894] |
carbonic anhydrase 7 in Human [GtoPdb: 2749] [UniProtKB: P43166] | ||||||||
GtoPdb | - | - | 8.68 | pKi | 2.1 | nM | Ki | Bioorg. Med. Chem. (2013) 21: 5973-82 [PMID:23965175] |
ChEMBL data shown on this page come from version 27:
Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]