ChEMBL ligand: CHEMBL783 (Starlix, DJN-608, Nateglinide, AY4166, AY-4166, SDZ DJN 608, A-4166, SDZ-DJN-608, Starsis, DJN 608)
Peptide transporter 2/Oligopeptide transporter, kidney isoform in Rat [ChEMBL: CHEMBL3325] [GtoPdb: 985] [UniProtKB: Q63424] This target only has 0 pki data point 0 1 CHEMBL783_lig_chart_1 Oligopeptide transporter, kidney isoform Rat There should be some charts here, you may need to enable JavaScript!
Organic anion transporter 1/Solute carrier family 22 member 6 in Rat [ChEMBL: CHEMBL1777665] [GtoPdb: 1025] [UniProtKB: O35956] 5.04 2 CHEMBL783_lig_chart_2 Solute carrier family 22 member 6 Rat There should be some charts here, you may need to enable JavaScript!

DB	Assay description	Assay Type	Standard value	Standard parameter	Original value	Original units	Original parameter	Reference
Peptide transporter 2/Oligopeptide transporter, kidney isoform in Rat (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3325] [GtoPdb: 985] [UniProtKB: Q63424]
ChEMBL	TP_TRANSPORTER: inhibition of Gly-Sar uptake (Gly-Sar: 20 uM) in PEPT2-expressing LLC-PK1 cells	F	4.15	pIC50	70000	nM	IC50	Eur. J. Pharmacol. (2000) 392: 11-17 [PMID:10748266]
Organic anion transporter 1/Solute carrier family 22 member 6 in Rat (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL1777665] [GtoPdb: 1025] [UniProtKB: O35956]
ChEMBL	Inhibition of rat Oat1 expressed in Xenopus oocytes	B	5.04	pKi	9200	nM	Ki	Bioorg. Med. Chem. (2011) 19: 3320-3340 [PMID:21571536]
ChEMBL	TP_TRANSPORTER: inhibition of PAH uptake in Xenopus laevis oocytes	F	5.04	pKi	9200	nM	Ki	Eur. J. Pharmacol. (2000) 398: 193-197 [PMID:10854830]

ChEMBL data shown on this page come from version 28:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]