adrenomedullin 2/intermedin | Ligand Activity Charts | IUPHAR/BPS Guide to PHARMACOLOGY

adrenomedullin 2/intermedin [Ligand Id: 684] activity data from GtoPdb

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CT receptor in Human [GtoPdb: 43] [UniProtKB: P30988] There should be some charts here, you may need to enable JavaScript!
AMY₁ receptor in Human [GtoPdb: 44] There should be some charts here, you may need to enable JavaScript!
AMY₂ receptor in Human [GtoPdb: 45] There should be some charts here, you may need to enable JavaScript!
AMY₃ receptor in Human [GtoPdb: 46] There should be some charts here, you may need to enable JavaScript!
CGRP receptor in Human [GtoPdb: 48] There should be some charts here, you may need to enable JavaScript!
AM₁ receptor in Human [GtoPdb: 49] There should be some charts here, you may need to enable JavaScript!
AM₂ receptor in Human [GtoPdb: 50] There should be some charts here, you may need to enable JavaScript!

DB	Assay description	Assay Type	Standard value	Standard parameter	Original value	Original units	Original parameter	Reference
CT receptor in Human [GtoPdb: 43] [UniProtKB: P30988]
GtoPdb	-	-	6.5	pEC50	-	-	-	Mol Pharmacol (2005) 67: 1655-65 [PMID:15692146]
AMY₁ receptor in Human [GtoPdb: 44]
GtoPdb	-	-	8	pEC50	-	-	-	Br J Pharmacol (2012) 166: 110-20 [PMID:21658025]
AMY₂ receptor in Human [GtoPdb: 45]
GtoPdb	-	-	6	pEC50	-	-	-	Br J Pharmacol (2012) 166: 110-20 [PMID:21658025]
AMY₃ receptor in Human [GtoPdb: 46]
GtoPdb	-	-	7	pEC50	-	-	-	Br J Pharmacol (2012) 166: 110-20 [PMID:21658025]
CGRP receptor in Human [GtoPdb: 48]
GtoPdb	-	-	9.1	pEC50	-	-	-	Br J Pharmacol (2012) 166: 110-20 [PMID:21658025]
AM₁ receptor in Human [GtoPdb: 49]
GtoPdb	-	-	8.3	pEC50	-	-	-	Br J Pharmacol (2018) 175: 3-17 [PMID:29059473]
AM₂ receptor in Human [GtoPdb: 50]
GtoPdb	-	-	10.1	pEC50	-	-	-	Br J Pharmacol (2018) 175: 3-17 [PMID:29059473]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.