amylin [Ligand Id: 688] activity data from GtoPdb

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  • CT receptor in Human [GtoPdb: 43] [UniProtKB: P30988]
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  • AMY1 receptor in Human [GtoPdb: 44]
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  • AMY2 receptor in Human [GtoPdb: 45]
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  • AMY3 receptor in Human [GtoPdb: 46]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
CT receptor in Human [GtoPdb: 43] [UniProtKB: P30988]
GtoPdb - - 9.5 pEC50 - - - Mol. Pharmacol. (2005) 67: 1655-65 [PMID:15692146];
J. Endocrinol. (1997) 155: 423-31 [PMID:9487987];
J Pharmacol Toxicol Methods (1999) 42: 217-24 [PMID:11033437]
AMY1 receptor in Human [GtoPdb: 44]
GtoPdb - - 10.7 pEC50 0.02 nM EC50 Mol. Pharmacol. (2005) 67: 1655-65 [PMID:15692146];
Mol. Pharmacol. (2004) 65: 207-13 [PMID:14722252];
J Pharmacol Toxicol Methods (1999) 42: 217-24 [PMID:11033437];
Endocrinology (2014) 155: 21-6 [PMID:24169554]
AMY2 receptor in Human [GtoPdb: 45]
GtoPdb - - 9.9 pEC50 0.13 nM EC50 Mol. Pharmacol. (2004) 65: 207-13 [PMID:14722252];
J Pharmacol Toxicol Methods (1999) 42: 217-24 [PMID:11033437];
Endocrinology (2014) 155: 21-6 [PMID:24169554]
AMY3 receptor in Human [GtoPdb: 46]
GtoPdb - - 10.8 pEC50 - - - Mol. Pharmacol. (2005) 67: 1655-65 [PMID:15692146];
J Pharmacol Toxicol Methods (1999) 42: 217-24 [PMID:11033437];
Endocrinology (2014) 155: 21-6 [PMID:24169554]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.