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ChEMBL ligand: CHEMBL464925 ((8E,11E,14E)-Anacardic Acid) |
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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Glyceraldehyde-3-phosphate dehydrogenase, glycosomal in Trypanosoma cruzi (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL5926] [UniProtKB: P22513] | ||||||||
ChEMBL | Inhibition of Trypanosoma cruzi recombinant glycosomal GAPDH expressed in Escherichia coli by spectrophotometry | B | 4.42 | pIC50 | 38000 | nM | IC50 | Bioorg Med Chem (2009) 17: 2476-2482 [PMID:19254846] |
E1A binding protein p300 in Human [GtoPdb: 2735] [UniProtKB: Q09472] | ||||||||
GtoPdb | - | - | 5.3 | pIC50 | 5000 | nM | IC50 | J Biol Chem (2003) 278: 19134-40 [PMID:12624111] |
lysine acetyltransferase 2B in Human [GtoPdb: 2737] [UniProtKB: Q92831] | ||||||||
GtoPdb | - | - | 5.07 | pIC50 | 8500 | nM | IC50 |
ChEMBL data shown on this page come from version 32:
Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]