anacardic acid [Ligand Id: 6999] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL464925 ((8E,11E,14E)-Anacardic Acid)
  • Glyceraldehyde-3-phosphate dehydrogenase, glycosomal in Trypanosoma cruzi [ChEMBL: CHEMBL5926] [UniProtKB: P22513]
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  • E1A binding protein p300 in Human [GtoPdb: 2735] [UniProtKB: Q09472]
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  • lysine acetyltransferase 2B in Human [GtoPdb: 2737] [UniProtKB: Q92831]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Glyceraldehyde-3-phosphate dehydrogenase, glycosomal in Trypanosoma cruzi (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL5926] [UniProtKB: P22513]
ChEMBL Inhibition of Trypanosoma cruzi recombinant glycosomal GAPDH expressed in Escherichia coli by spectrophotometry B 4.42 pIC50 38000 nM IC50 Bioorg. Med. Chem. (2009) 17: 2476-2482 [PMID:19254846]
E1A binding protein p300 in Human [GtoPdb: 2735] [UniProtKB: Q09472]
GtoPdb - - 5.3 pIC50 5000 nM IC50 J. Biol. Chem. (2003) 278: 19134-40 [PMID:12624111]
lysine acetyltransferase 2B in Human [GtoPdb: 2737] [UniProtKB: Q92831]
GtoPdb - - 5.07 pIC50 8500 nM IC50

ChEMBL data shown on this page come from version 27:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]