H3-CoA-20 [Ligand Id: 7035] activity data from GtoPdb and ChEMBL

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

ChEMBL ligand: CHEMBL1221562
  • E1A binding protein p300 in Human [GtoPdb: 2735] [UniProtKB: Q09472]
There should be some charts here, you may need to enable JavaScript!
  • lysine acetyltransferase 2B in Human [GtoPdb: 2737] [UniProtKB: Q92831]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
E1A binding protein p300 in Human [GtoPdb: 2735] [UniProtKB: Q09472]
GtoPdb - - 3.7 pIC50 200000 nM IC50 Mol Cell (2000) 5: 589-95 [PMID:10882143]
lysine acetyltransferase 2B in Human [GtoPdb: 2737] [UniProtKB: Q92831]
GtoPdb - - 6.52 pIC50 300 nM IC50 Mol Cell (2000) 5: 589-95 [PMID:10882143]

ChEMBL data shown on this page come from version 33:

Mendez D, Gaulton A, Bento AP, Chambers J, De Veij M, Félix E, Magariños MP, Mosquera JF, Mutowo P, Nowotka M, Gordillo-Marañón M, Hunter F, Junco L, Mugumbate G, Rodriguez-Lopez M, Atkinson F, Bosc N, Radoux CJ, Segura-Cabrera A, Hersey A, Leach AR. (2019) 'ChEMBL: towards direct deposition of bioassay data' Nucleic Acids Res., 47(D1). DOI: 10.1093/nar/gky1075. [EPMCID:30398643]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]