H3-CoA-20 [Ligand Id: 7035] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL1221562
  • E1A binding protein p300 in Human [GtoPdb: 2735] [UniProtKB: Q09472]
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  • lysine acetyltransferase 2B in Human [GtoPdb: 2737] [UniProtKB: Q92831]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
E1A binding protein p300 in Human [GtoPdb: 2735] [UniProtKB: Q09472]
GtoPdb - - 3.7 pIC50 200000 nM IC50 Mol Cell (2000) 5: 589-95 [PMID:10882143]
lysine acetyltransferase 2B in Human [GtoPdb: 2737] [UniProtKB: Q92831]
GtoPdb - - 6.52 pIC50 300 nM IC50 Mol Cell (2000) 5: 589-95 [PMID:10882143]

ChEMBL data shown on this page come from version 28:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]