ChEMBL ligand: CHEMBL799 (Pletal, OPC-13013, Cilostazol, OPC-21)
CYP2C9/Cytochrome P450 2C9 in Human [ChEMBL: CHEMBL3397] [GtoPdb: 1326] [UniProtKB: P11712] This target only has 0 pki data point 1 CHEMBL799_lig_chart_1 Cytochrome P450 2C9 Human There should be some charts here, you may need to enable JavaScript!
Plasmodium falciparum [ChEMBL: CHEMBL364] This target only has 0 pki data point 2 CHEMBL799_lig_chart_2 Plasmodium falciparum Plasmodium falciparum There should be some charts here, you may need to enable JavaScript!
phosphodiesterase 3A in Human [GtoPdb: 1298] [UniProtKB: Q14432] This target only has 0 pki data point 3 CHEMBL799_lig_chart_3 phosphodiesterase 3A Human There should be some charts here, you may need to enable JavaScript!
phosphodiesterase 3B in Human [GtoPdb: 1299] [UniProtKB: Q13370] This target only has 0 pki data point 4 CHEMBL799_lig_chart_4 phosphodiesterase 3B Human There should be some charts here, you may need to enable JavaScript!

DB	Assay description	Assay Type	Standard value	Standard parameter	Original value	Original units	Original parameter	Reference
CYP2C9/Cytochrome P450 2C9 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL3397] [GtoPdb: 1326] [UniProtKB: P11712]
ChEMBL	DRUGMATRIX: CYP450, 2C9 enzyme inhibition (substrate: 3-Cyano-7-ethoxycoumarin)	B	5	pIC50	10000	nM	IC50	DrugMatrix in vitro pharmacology data
Plasmodium falciparum (target type: ORGANISM) [ChEMBL: CHEMBL364]
ChEMBL	Antiplasmodial activity against Plasmodium falciparum 3D7 after 72 hrs by SYBR green assay	F	4.9	pIC50	12589.25	nM	IC50	Nat. Chem. Biol. (2009) 5: 765-771 [PMID:19734910]
ChEMBL	Antiplasmodial activity against Plasmodium falciparum HB3 after 72 hrs by SYBR green assay	F	4.9	pIC50	12589.25	nM	IC50	Nat. Chem. Biol. (2009) 5: 765-771 [PMID:19734910]
ChEMBL	Antiplasmodial activity against Plasmodium falciparum 7G8 after 72 hrs by SYBR green assay	F	5	pIC50	10000	nM	IC50	Nat. Chem. Biol. (2009) 5: 765-771 [PMID:19734910]
ChEMBL	Antiplasmodial activity against Plasmodium falciparum D10 after 72 hrs by SYBR green assay	F	5	pIC50	10000	nM	IC50	Nat. Chem. Biol. (2009) 5: 765-771 [PMID:19734910]
ChEMBL	Antiplasmodial activity against Plasmodium falciparum W2 after 72 hrs by SYBR green assay	F	5	pIC50	10000	nM	IC50	Nat. Chem. Biol. (2009) 5: 765-771 [PMID:19734910]
phosphodiesterase 3A in Human [GtoPdb: 1298] [UniProtKB: Q14432]
GtoPdb	-	-	6.7	pIC50	200	nM	IC50	Biochem. Pharmacol. (2000) 59: 347-56 [PMID:10644042]
phosphodiesterase 3B in Human [GtoPdb: 1299] [UniProtKB: Q13370]
GtoPdb	-	-	6.42	pIC50	380	nM	IC50	Biochem. Pharmacol. (2000) 59: 347-56 [PMID:10644042]

ChEMBL data shown on this page come from version 27:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]