alimemazine [Ligand Id: 7237] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL829 (Alimemazine, BAYER-1219, Dl-trimeprazine, Methylpromazine, RP-6549, Temaril, Trimeprazine)
  • H1 receptor in Bovine [GtoPdb: 262]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
H1 receptor in Bovine [GtoPdb: 262]
GtoPdb Inhibition of [3H]mepyramine binding to bovine brain membrane preparations in vitro. - 9.14 pKi 0.72 nM Ki Jpn J Pharmacol (1987) 43: 277-82 [PMID:2884340]

ChEMBL data shown on this page come from version 31:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]