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ChEMBL ligand: CHEMBL829 (Alimemazine, BAYER-1219, Dl-trimeprazine, Methylpromazine, RP-6549, Temaril, Trimeprazine) |
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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H1 receptor in Bovine [GtoPdb: 262] | ||||||||
GtoPdb | Inhibition of [3H]mepyramine binding to bovine brain membrane preparations in vitro. | - | 9.14 | pKi | 0.72 | nM | Ki | Jpn J Pharmacol (1987) 43: 277-82 [PMID:2884340] |
ChEMBL data shown on this page come from version 31:
Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]