lixisenatide [Ligand Id: 7387] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL2108336 (ZP-10, Lyxumia, Lixisenatide, ZP 10, AVE0010, AVE 010, Adlyxin, AVE-0010, AVE-010)
  • GLP-1 receptor in Human [GtoPdb: 249] [UniProtKB: P43220]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
GLP-1 receptor in Human [GtoPdb: 249] [UniProtKB: P43220]
GtoPdb CHO-K1 cells overexpressing the human GLP-1 receptor. - 8.88 pKi 1.33 nM Ki Regul Pept (2010) 164: 58-64 [PMID:20570597]

ChEMBL data shown on this page come from version 28:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, Cibrián-Uhalte E, Davies M, Dedman N, Karlsson A, Magariños MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]