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ChEMBL ligand: CHEMBL2108184 (Crofelemer, Fulyzaq, Mytesi, NP-303, Provir, SP-303, TRN-002, Virend) |
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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CFTR in Human [GtoPdb: 707] [UniProtKB: P13569] | ||||||||
GtoPdb | - | - | 5.15 | pIC50 | 7000 | nM | IC50 | Mol Pharmacol (2010) 77: 69-78 [PMID:19808995] |
CaCC in Human [GtoPdb: 708] [UniProtKB: Q5XXA6] | ||||||||
GtoPdb | - | - | 5.19 | pIC50 | 6500 | nM | IC50 | Mol Pharmacol (2010) 77: 69-78 [PMID:19808995] |
ChEMBL data shown on this page come from version 31:
Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]