protoxin II [Ligand Id: 7571] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • Nav1.2 in Human [GtoPdb: 579] [UniProtKB: Q99250]
There should be some charts here, you may need to enable JavaScript!
  • Nav1.5 in Human [GtoPdb: 582] [UniProtKB: Q14524]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Nav1.2 in Human [GtoPdb: 579] [UniProtKB: Q99250]
GtoPdb Whole cell voltage clamp of transfected human embryonic kidney cells (HEK293) - 7.4 pKi - - - Mol Pharmacol (2008) 74: 1476-84 [PMID:18728100]
Nav1.5 in Human [GtoPdb: 582] [UniProtKB: Q14524]
GtoPdb Whole-cell voltage clamp of human Nav1.5 channels expressed in human embryonic kidney cells (HEK293). - 6.5 pKi - - - Biochemistry (2002) 41: 14734-47 [PMID:12475222]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.