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1
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CCR1
Human
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2
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CCR2
Human
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3
_lig_chart_3
CCR3
Human
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4
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CCR5
Human
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5
_lig_chart_5
CXCR3
Human
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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CCR1 in Human [GtoPdb: 58] [UniProtKB: P32246] | ||||||||
GtoPdb | - | - | 8.1 | pKi | - | - | - |
Br. J. Pharmacol. (2002) 137: 663-75 [PMID:12381680]; Mol. Hum. Reprod. (2002) 8: 419-25 [PMID:11994538] |
CCR2 in Human [GtoPdb: 59] [UniProtKB: P41597] | ||||||||
GtoPdb | - | - | 8.7 | pIC50 | - | - | - |
J. Clin. Invest. (1997) 100: 1137-43 [PMID:9276730]; Eur. J. Biochem. (1997) 248: 507-15 [PMID:9346309]; J. Biol. Chem. (2003) 278: 10928-33 [PMID:12554737] |
CCR3 in Human [GtoPdb: 60] [UniProtKB: P51677] | ||||||||
GtoPdb | - | - | 9.2 | pKi | - | - | - | J. Exp. Med. (1996) 183: 2349-54 [PMID:8642344] |
CCR5 in Human [GtoPdb: 62] [UniProtKB: P51681] | ||||||||
GtoPdb | - | - | 7.5 | pKi | - | - | - | Biochem. Pharmacol. (2005) 71: 163-72 [PMID:16298345] |
CXCR3 in Human [GtoPdb: 70] [UniProtKB: P49682] | ||||||||
GtoPdb | - | - | 6.6 | pKi | - | - | - | J. Biol. Chem. (1998) 273: 18288-91 [PMID:9660793] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.