ABT-639 [Ligand Id: 7721] activity data from GtoPdb

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  • Cav3.1 in Human [GtoPdb: 535] [UniProtKB: O43497]
  • This target only has 0 pki data point
  • 0
1 _lig_chart_1 Cav3.1 Human
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  • Cav3.2 in Human [GtoPdb: 536] [UniProtKB: O95180]
  • This target only has 0 pki data point
  • 0
2 _lig_chart_2 Cav3.2 Human
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  • Cav3.3 in Human [GtoPdb: 537] [UniProtKB: Q9P0X4]
  • This target only has 0 pki data point
  • 0
3 _lig_chart_3 Cav3.3 Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Cav3.1 in Human [GtoPdb: 535] [UniProtKB: O43497]
GtoPdb - - 5 pIC50 - - - Biochem Pharmacol (2014) 89: 536-44 [PMID:24726441]
Cav3.2 in Human [GtoPdb: 536] [UniProtKB: O95180]
GtoPdb - - 5.6 pIC50 - - - Biochem Pharmacol (2014) 89: 536-44 [PMID:24726441]
Cav3.3 in Human [GtoPdb: 537] [UniProtKB: Q9P0X4]
GtoPdb - - 5 pIC50 - - - Biochem Pharmacol (2014) 89: 536-44 [PMID:24726441]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.