DQP-1105 [Ligand Id: 7843] activity data from GtoPdb

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  • GluN2B in Rat [GtoPdb: 457] [UniProtKB: Q00960]
  • This target only has 0 pki data point
  • 0
1 _lig_chart_1 GluN2B Rat
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  • GluN2C in Rat [GtoPdb: 458] [UniProtKB: Q00961]
  • This target only has 0 pki data point
  • 0
2 _lig_chart_2 GluN2C Rat
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  • GluN2D in Rat [GtoPdb: 459] [UniProtKB: Q62645]
  • This target only has 0 pki data point
  • 0
3 _lig_chart_3 GluN2D Rat
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
GluN2B in Rat [GtoPdb: 457] [UniProtKB: Q00960]
GtoPdb Measured using recombinant GluN1-1a NMDA subunits co-expressed with GluN2C subunits. - 6.95 pIC50 113 nM IC50 Mol Pharmacol (2011) 80: 782-95 [PMID:21807990]
GluN2C in Rat [GtoPdb: 458] [UniProtKB: Q00961]
GtoPdb Measured using recombinant GluN1-1a NMDA subunits co-expressed with GluN2C subunits. - 8.15 pIC50 7 nM IC50 Mol Pharmacol (2011) 80: 782-95 [PMID:21807990]
GluN2D in Rat [GtoPdb: 459] [UniProtKB: Q62645]
GtoPdb Measured using recombinant GluN1-1a NMDA subunits co-expressed with GluN2D subunits. - 5.57 pIC50 2700 nM IC50 Mol Pharmacol (2011) 80: 782-95 [PMID:21807990]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.