AKN-028 [Ligand Id: 7969] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| KIT proto-oncogene, receptor tyrosine kinase in Human [GtoPdb: 1805] [UniProtKB: P10721] | ||||||||
| GtoPdb | Inhibition of KIT autophosphorylation in human AML M07 cells which overexpress KIT | - | 7.54 | pIC50 | 29 | nM | IC50 | Blood Cancer J (2012) 2: e81 [PMID:22864397] |
| fms related receptor tyrosine kinase 3 in Human [GtoPdb: 1807] [UniProtKB: P36888] | ||||||||
| GtoPdb | - | - | 8.22 | pIC50 | 6 | nM | IC50 | Blood Cancer J (2012) 2: e81 [PMID:22864397] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
