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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| C-terminal Src kinase in Human [GtoPdb: 1994] [UniProtKB: P41240] | ||||||||
| GtoPdb | - | - | 7.25 | pIC50 | 56.4 | nM | IC50 | J Med Chem (2015) 58: 183-96 [PMID:25075558] |
| LYN proto-oncogene, Src family tyrosine kinase in Human [GtoPdb: 2060] [UniProtKB: P07948] | ||||||||
| GtoPdb | - | - | 7.89 | pIC50 | 12.9 | nM | IC50 | J Med Chem (2015) 58: 183-96 [PMID:25075558] |
| mitogen-activated protein kinase kinase kinase 7 in Human [GtoPdb: 2082] [UniProtKB: O43318] | ||||||||
| GtoPdb | - | - | 6.83 | pIC50 | 149 | nM | IC50 | J Med Chem (2015) 58: 183-96 [PMID:25075558] |
| mitogen-activated protein kinase kinase kinase kinase 2 in Human [GtoPdb: 2086] [UniProtKB: Q12851] | ||||||||
| GtoPdb | - | - | 7.66 | pIC50 | 21.7 | nM | IC50 | J Med Chem (2015) 58: 183-96 [PMID:25075558] |
| SRC proto-oncogene, non-receptor tyrosine kinase in Human [GtoPdb: 2206] [UniProtKB: P12931] | ||||||||
| GtoPdb | - | - | 6.95 | pIC50 | 113 | nM | IC50 | J Med Chem (2015) 58: 183-96 [PMID:25075558] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.