compound 27 [PMID: 18337095] [Ligand Id: 8158] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL255607
  • calcium/calmodulin-dependent protein kinase II delta subunit/CaM kinase II delta in Human [ChEMBL: CHEMBL2801] [GtoPdb: 1558] [UniProtKB: Q13557]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
calcium/calmodulin-dependent protein kinase II delta subunit/CaM kinase II delta in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL2801] [GtoPdb: 1558] [UniProtKB: Q13557]
GtoPdb - - 8 pIC50 10 nM IC50 Bioorg. Med. Chem. Lett. (2008) 18: 2399-403 [PMID:18337095]
ChEMBL Inhibition of CaMK2delta B 8 pIC50 10 nM IC50 Bioorg. Med. Chem. Lett. (2008) 18: 2399-2403 [PMID:18337095]

ChEMBL data shown on this page come from version 27:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]