Click here for a description of the charts and data table
Please tell us if you are using this feature and what you think!
|
There should be some charts here, you may need to enable JavaScript!
|
|
There should be some charts here, you may need to enable JavaScript!
|
| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| CXCR1 in Human [GtoPdb: 68] [UniProtKB: P25024] | ||||||||
| GtoPdb | - | - | 8.1 | pKd | 8 | nM | Kd | Blood (2012) 119: 2274-83 [PMID:22262769] |
| GtoPdb | - | - | 9.5 | pKi | - | - | - |
J Biol Chem (1992) 267: 16283-7 [PMID:1379593]; Br J Pharmacol (1999) 126: 810-8 [PMID:10188995]; J Biol Chem (2005) 280: 28663-74 [PMID:15946947]; J Biol Chem (1996) 271: 31202-9 [PMID:8940121]; Proc Natl Acad Sci USA (2004) 101: 11791-6 [PMID:15282370] |
| CXCR2 in Human [GtoPdb: 69] [UniProtKB: P25025] | ||||||||
| GtoPdb | - | - | 9.5 | pKi | - | - | - |
J Biol Chem (1992) 267: 16283-7 [PMID:1379593]; Br J Pharmacol (1999) 126: 810-8 [PMID:10188995]; J Biol Chem (2005) 280: 28663-74 [PMID:15946947]; J Biol Chem (1996) 271: 31202-9 [PMID:8940121]; Proc Natl Acad Sci USA (2004) 101: 11791-6 [PMID:15282370] |
| CXCR2 in Mouse [GtoPdb: 69] [UniProtKB: P35343] | ||||||||
| GtoPdb | - | - | 6.4 | pKi | - | - | - | J Biol Chem (1994) 269: 29355-8 [PMID:7961909] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.