GSK2801 [Ligand Id: 8233] activity data from GtoPdb

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  • bromodomain adjacent to zinc finger domain 2A in Human [GtoPdb: 2721] [UniProtKB: Q9UIF9]
  • This target only has 0 pki data point
1 _lig_chart_1 bromodomain adjacent to zinc finger domain 2A Human
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  • bromodomain adjacent to zinc finger domain 2B in Human [GtoPdb: 2722] [UniProtKB: Q9UIF8]
  • This target only has 0 pki data point
2 _lig_chart_2 bromodomain adjacent to zinc finger domain 2B Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
bromodomain adjacent to zinc finger domain 2A in Human [GtoPdb: 2721] [UniProtKB: Q9UIF9]
GtoPdb Isothermal titration calorimetry (ITC) assay - 6.59 pKd 257 nM Kd GSK2801: A Selective Chemical Probe for BAZ2B/A bromodomains.. thesgc.org
bromodomain adjacent to zinc finger domain 2B in Human [GtoPdb: 2722] [UniProtKB: Q9UIF8]
GtoPdb Isothermal titration calorimetry (ITC) assay - 6.87 pKd 136 nM Kd GSK2801: A Selective Chemical Probe for BAZ2B/A bromodomains.. thesgc.org

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.