[125I]BH-MIT1 [Ligand Id: 8522] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • PKR1 in Human [GtoPdb: 335] [UniProtKB: Q8TCW9]
There should be some charts here, you may need to enable JavaScript!
  • PKR2 in Human [GtoPdb: 336] [UniProtKB: Q8NFJ6]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
PKR1 in Human [GtoPdb: 335] [UniProtKB: Q8TCW9]
GtoPdb - - 8.39 pIC50 4.1 nM IC50 Biochem Biophys Res Commun (2002) 293: 396-402 [PMID:12054613]
PKR2 in Human [GtoPdb: 336] [UniProtKB: Q8NFJ6]
GtoPdb - - 9.17 pIC50 0.67 nM IC50 Biochem Biophys Res Commun (2002) 293: 396-402 [PMID:12054613]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.