NI-57 [Ligand Id: 8573] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| bromodomain containing 1 in Human [GtoPdb: 2724] [UniProtKB: O95696] | ||||||||
| GtoPdb | - | - | 6.97 | pKd | 108 | nM | Kd | NI-57 – a chemical probe for BRPF bromodomains.. thesgc.org |
| bromodomain and PHD finger containing 1 in Human [GtoPdb: 2730] [UniProtKB: P55201] | ||||||||
| GtoPdb | Isothermal titration calorimetry (ITC) assay, measuring binding to BRPF1B isoform. | - | 7.51 | pKd | 31 | nM | Kd | NI-57 – a chemical probe for BRPF bromodomains.. thesgc.org |
| bromodomain and PHD finger containing 3 in Human [GtoPdb: 2731] [UniProtKB: Q9ULD4] | ||||||||
| GtoPdb | - | - | 6.39 | pKd | 408 | nM | Kd | NI-57 – a chemical probe for BRPF bromodomains.. thesgc.org |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
