Alexa-488-telenzepine [Ligand Id: 8600] activity data from GtoPdb

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  • M1 receptor in Human [GtoPdb: 13] [UniProtKB: P11229]
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  • M2 receptor in Human [GtoPdb: 14] [UniProtKB: P08172]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
M1 receptor in Human [GtoPdb: 13] [UniProtKB: P11229]
GtoPdb - - 9.3 pKd - - - Proc. Natl. Acad. Sci. U.S.A. (2010) 107: 2693-8 [PMID:20133736]
M2 receptor in Human [GtoPdb: 14] [UniProtKB: P08172]
GtoPdb - - 8.8 pKi - - - J. Mol. Cell. Cardiol. (2013) 57: 129-36 [PMID:23357106]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.