compound 16 [PMID: 19097778] [Ligand Id: 8837] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL482331
  • Solute carrier family 28 member 3 in Human [ChEMBL: CHEMBL5707] [GtoPdb: 1116] [UniProtKB: Q9HAS3]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Solute carrier family 28 member 3 in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL5707] [GtoPdb: 1116] [UniProtKB: Q9HAS3]
GtoPdb - - 5.54 pKi 2880 nM Ki Bioorg Med Chem Lett (2009) 19: 917-21 [PMID:19097778]
ChEMBL Binding affinity to human recombinant CNT3 expressed in pig PK15NTD cells assessed as [3H]uridine uptake by beta-scintillation counter B 5.54 pKi 2880 nM Ki Bioorg. Med. Chem. Lett. (2009) 19: 917-921 [PMID:19097778]

ChEMBL data shown on this page come from version 28:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]