4-acryloylphenol [Ligand Id: 8841] activity data from GtoPdb and ChEMBL
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| ChEMBL ligand: CHEMBL378577 (4-Acryloylphenol) |
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| 4-aminobutyrate aminotransferase/Gamma-amino-N-butyrate transaminase in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL2044] [GtoPdb: 2464] [UniProtKB: P80404] | ||||||||
| GtoPdb | - | - | 5.26 | pIC50 | 5480 | nM | IC50 | Bioorg Med Chem Lett (2006) 16: 592-5 [PMID:16290145] |
| ChEMBL | Inhibitory activity against GABAT | B | 5.26 | pIC50 | 5480 | nM | IC50 | Bioorg Med Chem Lett (2006) 16: 592-595 [PMID:16290145] |
| aldehyde dehydrogenase 5 family member A1/Succinate semialdehyde dehydrogenase in Human (target type: SINGLE PROTEIN) [ChEMBL: CHEMBL1911] [GtoPdb: 2466] [UniProtKB: P51649] | ||||||||
| ChEMBL | Inhibitory activity against SSADH | B | 6.46 | pIC50 | 350 | nM | IC50 | Bioorg Med Chem Lett (2006) 16: 592-595 [PMID:16290145] |
| GtoPdb | - | - | 6.46 | pIC50 | 350 | nM | IC50 | Bioorg Med Chem Lett (2006) 16: 592-5 [PMID:16290145] |
ChEMBL data shown on this page come from version 34:
Zdrazil B, Felix E, Hunter F, Manners EJ, Blackshaw J, Corbett S, de Veij M, Ioannidis H, Lopez DM, Mosquera JF, Magarinos MP, Bosc N, Arcila R, Kizilören T, Gaulton A, Bento AP, Adasme MF, Monecke P, Landrum GA, Leach AR. (2024). The ChEMBL Database in 2023: a drug discovery platform spanning multiple bioactivity data types and time periods. Nucleic Acids Res., 52(D1). DOI: 10.1093/nar/gkad1004. [EPMCID:10767899] [PMID:37933841]
Davies M, Nowotka M, Papadatos G, Dedman N, Gaulton A, Atkinson F, Bellis L, Overington JP. (2015) 'ChEMBL web services: streamlining access to drug discovery data and utilities.' Nucleic Acids Res., 43(W1). DOI: 10.1093/nar/gkv352. [EPMCID:25883136]
