AT-076 [Ligand Id: 8870] activity data from GtoPdb

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  • δ receptor in Human [GtoPdb: 317] [UniProtKB: P41143]
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  • κ receptor in Human [GtoPdb: 318] [UniProtKB: P41145]
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  • μ receptor in Human [GtoPdb: 319] [UniProtKB: P35372]
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  • NOP receptor in Human [GtoPdb: 320] [UniProtKB: P41146]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
δ receptor in Human [GtoPdb: 317] [UniProtKB: P41143]
GtoPdb Radioligand binding assay - 7.71 pKi 19.6 nM Ki NIDA Res Monogr (1998) 178: 440-66 [PMID:9686407];
Life Sci (2003) 73: 663-678 [PMID:12801588]
κ receptor in Human [GtoPdb: 318] [UniProtKB: P41145]
GtoPdb Radioligand binding assay - 8.94 pKi 1.14 nM Ki NIDA Res Monogr (1998) 178: 440-66 [PMID:9686407];
ACS Chem Neurosci (2015) 6: 646-57 [PMID:25635572]
μ receptor in Human [GtoPdb: 319] [UniProtKB: P35372]
GtoPdb Radioligand binding assay - 8.78 pKi 1.67 nM Ki NIDA Res Monogr (1998) 178: 440-66 [PMID:9686407];
ACS Chem Neurosci (2015) 6: 646-57 [PMID:25635572]
NOP receptor in Human [GtoPdb: 320] [UniProtKB: P41146]
GtoPdb Radioligand binding assay - 8.76 pKi 1.75 nM Ki ACS Chem Neurosci (2015) 6: 646-57 [PMID:25635572]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.