AC-186 [Ligand Id: 8897] activity data from GtoPdb

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  • Estrogen receptor-α in Human [GtoPdb: 620] [UniProtKB: P03372]
  • This target only has 0 pki data point
  • 0
1 _lig_chart_1 Estrogen receptor-α Human
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  • Estrogen receptor-β in Human [GtoPdb: 621] [UniProtKB: Q92731]
  • This target only has 0 pki data point
  • 0
2 _lig_chart_2 Estrogen receptor-β Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Estrogen receptor-α in Human [GtoPdb: 620] [UniProtKB: P03372]
GtoPdb Measured using Receptor Selection and Amplification Technology (R-SAT). - 5.3 pEC50 5000 nM EC50 ACS Chem Neurosci (2013) 4: 1249-55 [PMID:23898966]
Estrogen receptor-β in Human [GtoPdb: 621] [UniProtKB: Q92731]
GtoPdb Measured using Receptor Selection and Amplification Technology (R-SAT). - 8.22 pEC50 6 nM EC50 ACS Chem Neurosci (2013) 4: 1249-55 [PMID:23898966]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.