A-196 [Ligand Id: 8949] activity data from GtoPdb

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  • lysine methyltransferase 5B in Human [GtoPdb: 2717] [UniProtKB: Q4FZB7]
  • This target only has 0 pki data point
  • 0
1 _lig_chart_1 lysine methyltransferase 5B Human
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  • lysine methyltransferase 5C in Human [GtoPdb: 2718] [UniProtKB: Q86Y97]
  • This target only has 0 pki data point
  • 0
2 _lig_chart_2 lysine methyltransferase 5C Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
lysine methyltransferase 5B in Human [GtoPdb: 2717] [UniProtKB: Q4FZB7]
GtoPdb In vitro activity. - 7.6 pIC50 25 nM IC50 A-196 A selective chemical probe for SUV420H1/H2. The Structural Genomics Consortium
lysine methyltransferase 5C in Human [GtoPdb: 2718] [UniProtKB: Q86Y97]
GtoPdb In vitro activity. - 6.84 pIC50 144 nM IC50 A-196 A selective chemical probe for SUV420H1/H2. The Structural Genomics Consortium

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.