A-196 [Ligand Id: 8949] activity data from GtoPdb

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  • lysine methyltransferase 5B in Human [GtoPdb: 2717] [UniProtKB: Q4FZB7]
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  • lysine methyltransferase 5C in Human [GtoPdb: 2718] [UniProtKB: Q86Y97]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
lysine methyltransferase 5B in Human [GtoPdb: 2717] [UniProtKB: Q4FZB7]
GtoPdb In vitro activity. - 7.6 pIC50 25 nM IC50 A-196 A selective chemical probe for SUV420H1/H2. thesgc.org
lysine methyltransferase 5C in Human [GtoPdb: 2718] [UniProtKB: Q86Y97]
GtoPdb In vitro activity. - 6.84 pIC50 144 nM IC50 A-196 A selective chemical probe for SUV420H1/H2. thesgc.org

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.