conessine [Ligand Id: 8981] activity data from GtoPdb

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  • H1 receptor in Human [GtoPdb: 262] [UniProtKB: P35367]
  • This target only has 1 pki data point
  • 5
1 _lig_chart_1 H1 receptor Human
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  • H2 receptor in Human [GtoPdb: 263] [UniProtKB: P25021]
  • This target only has 1 pki data point
  • 5
2 _lig_chart_2 H2 receptor Human
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  • H3 receptor in Human [GtoPdb: 264] [UniProtKB: Q9Y5N1]
  • This target only has 1 pki data point
  • 8.3
3 _lig_chart_3 H3 receptor Human
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  • H4 receptor in Human [GtoPdb: 265] [UniProtKB: Q9H3N8]
  • This target only has 1 pki data point
  • 5
4 _lig_chart_4 H4 receptor Human
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
H1 receptor in Human [GtoPdb: 262] [UniProtKB: P35367]
GtoPdb - - 5 pKi >10000 nM Ki Pharmacol Rev (2015) 67: 601-55 [PMID:26084539]
H2 receptor in Human [GtoPdb: 263] [UniProtKB: P25021]
GtoPdb - - 5 pKi >10000 nM Ki Pharmacol Rev (2015) 67: 601-55 [PMID:26084539]
H3 receptor in Human [GtoPdb: 264] [UniProtKB: Q9Y5N1]
GtoPdb - - 8.3 pKi - - - Pharmacol Rev (2015) 67: 601-55 [PMID:26084539]
H4 receptor in Human [GtoPdb: 265] [UniProtKB: Q9H3N8]
GtoPdb - - 5 pKi >10000 nM Ki Pharmacol Rev (2015) 67: 601-55 [PMID:26084539]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.