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1
_lig_chart_1
H1 receptor
Human
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2
_lig_chart_2
H2 receptor
Human
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3
_lig_chart_3
H3 receptor
Human
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4
_lig_chart_4
H4 receptor
Human
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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
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H1 receptor in Human [GtoPdb: 262] [UniProtKB: P35367] | ||||||||
GtoPdb | - | - | 5 | pKi | >10000 | nM | Ki | Pharmacol Rev (2015) 67: 601-55 [PMID:26084539] |
H2 receptor in Human [GtoPdb: 263] [UniProtKB: P25021] | ||||||||
GtoPdb | - | - | 5 | pKi | >10000 | nM | Ki | Pharmacol Rev (2015) 67: 601-55 [PMID:26084539] |
H3 receptor in Human [GtoPdb: 264] [UniProtKB: Q9Y5N1] | ||||||||
GtoPdb | - | - | 8.3 | pKi | - | - | - | Pharmacol Rev (2015) 67: 601-55 [PMID:26084539] |
H4 receptor in Human [GtoPdb: 265] [UniProtKB: Q9H3N8] | ||||||||
GtoPdb | - | - | 5 | pKi | >10000 | nM | Ki | Pharmacol Rev (2015) 67: 601-55 [PMID:26084539] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.