opicapone [Ligand Id: 8988] activity data from GtoPdb

Click here for a description of the charts and data table

Please tell us if you are using this feature and what you think!

  • Catechol-O-methyltransferase in Human [GtoPdb: 2472] [UniProtKB: P21964]
  • Catechol-O-methyltransferase in Mouse [GtoPdb: 2472] [UniProtKB: O88587]
  • Catechol-O-methyltransferase in Rat [GtoPdb: 2472] [UniProtKB: P22734]
There should be some charts here, you may need to enable JavaScript!
DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
Catechol-O-methyltransferase in Human [GtoPdb: 2472] [UniProtKB: P21964]
GtoPdb - - 9 pKi 1 nM Ki J Med Chem (2014) 57: 5459-63 [PMID:24847974]
Catechol-O-methyltransferase in Mouse [GtoPdb: 2472] [UniProtKB: O88587]
GtoPdb - - 8.82 pKi 1.5 nM Ki J Med Chem (2014) 57: 5459-63 [PMID:24847974]
Catechol-O-methyltransferase in Rat [GtoPdb: 2472] [UniProtKB: P22734]
GtoPdb - - 8.82 pKi 1.5 nM Ki J Med Chem (2014) 57: 5459-63 [PMID:24847974]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.