acenocoumarol [Ligand Id: 9015] activity data from GtoPdb and ChEMBL

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ChEMBL ligand: CHEMBL397420 (Sinthrome, Acenocoumarol, Nicoumalone, Acenocoumarin)
  • vitamin K epoxide reductase complex subunit 1 in Rat [GtoPdb: 2645] [UniProtKB: Q6TEK4]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
vitamin K epoxide reductase complex subunit 1 in Rat [GtoPdb: 2645] [UniProtKB: Q6TEK4]
GtoPdb - - 6.11 pIC50 770 nM IC50 Bioorg. Med. Chem. (2007) 15: 2414-20 [PMID:17275317]

ChEMBL data shown on this page come from version 26:

Gaulton A, Hersey A, Nowotka M, Bento AP, Chambers J, Mendez D, Mutowo P, Atkinson F, Bellis LJ, CibriƔn-Uhalte E, Davies M, Dedman N, Karlsson A, MagariƱos MP, Overington JP, Papadatos G, Smit I, Leach AR. (2017) 'The ChEMBL database in 2017.' Nucleic Acids Res., 45(D1). DOI: 10.1093/nar/gkw1074. [PMCID:5210557]