sauvagine [Ligand Id: 918] activity data from GtoPdb

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  • CRF1 receptor in Human [GtoPdb: 212] [UniProtKB: P34998]
  • This target only has 0 pki data point
1 _lig_chart_1 CRF1 receptor Human
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  • CRF2 receptor in Human [GtoPdb: 213] [UniProtKB: Q13324]
  • CRF2 receptor in Mouse [GtoPdb: 213] [UniProtKB: Q60748]
  • CRF2 receptor in Rat [GtoPdb: 213] [UniProtKB: P47866]
  • This target only has 0 pki data point
2 _lig_chart_2 CRF2 receptor HumanMouseRat
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
CRF1 receptor in Human [GtoPdb: 212] [UniProtKB: P34998]
GtoPdb - - 9.2 pKd - - - J. Neurochem. (1997) 69: 1640-9 [PMID:9326293];
Biochem Pharmacol. (2004) 68: 1833-1844 [PMID:15450949];
J. Pharmacol. Exp. Ther. (2001) 296: 113-20 [PMID:11123370];
Endocrinology (1996) 137: 2167-70 [PMID:8612563];
Nature (1995) 378: 287-92 [PMID:7477349];
J. Pharmacol. Exp. Ther. (1999) 288: 729-34 [PMID:9918582]
CRF2 receptor in Human [GtoPdb: 213] [UniProtKB: Q13324]
GtoPdb - - 9.3 pKd - - - Biochem Pharmacol. (2004) 68: 1833-1844 [PMID:15450949];
J. Pharmacol. Exp. Ther. (2001) 296: 113-20 [PMID:11123370]
CRF2 receptor in Mouse [GtoPdb: 213] [UniProtKB: Q60748]
GtoPdb - - 8.7 pKd - - - Endocrinology (1996) 137: 2167-70 [PMID:8612563];
Nature (1995) 378: 287-92 [PMID:7477349];
J. Pharmacol. Exp. Ther. (1999) 288: 729-34 [PMID:9918582]
CRF2 receptor in Rat [GtoPdb: 213] [UniProtKB: P47866]
GtoPdb - - 8.8 pKd - - - Endocrinology (1996) 137: 2167-70 [PMID:8612563];
J. Pharmacol. Exp. Ther. (1999) 288: 729-34 [PMID:9918582]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.