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DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
---|---|---|---|---|---|---|---|---|
ABL proto-oncogene 1, non-receptor tyrosine kinase in Human [GtoPdb: 1923] [UniProtKB: P00519] | ||||||||
GtoPdb | - | - | 6.32 | pIC50 | 479 | nM | IC50 | J Med Chem (2016) 59: 4697-710 [PMID:27115835] |
BLK proto-oncogene, Src family tyrosine kinase in Human [GtoPdb: 1940] [UniProtKB: P51451] | ||||||||
GtoPdb | - | - | 8.27 | pIC50 | 5.4 | nM | IC50 | J Med Chem (2016) 59: 4697-710 [PMID:27115835] |
FGR proto-oncogene, Src family tyrosine kinase in Human [GtoPdb: 2024] [UniProtKB: P09769] | ||||||||
GtoPdb | - | - | 9.3 | pIC50 | <0.5 | nM | IC50 | J Med Chem (2016) 59: 4697-710 [PMID:27115835] |
fyn related Src family tyrosine kinase in Human [GtoPdb: 2025] [UniProtKB: P42685] | ||||||||
GtoPdb | - | - | 8.55 | pIC50 | 2.8 | nM | IC50 | J Med Chem (2016) 59: 4697-710 [PMID:27115835] |
FYN proto-oncogene, Src family tyrosine kinase in Human [GtoPdb: 2026] [UniProtKB: P06241] | ||||||||
GtoPdb | - | - | 8.68 | pIC50 | 2.1 | nM | IC50 | J Med Chem (2016) 59: 4697-710 [PMID:27115835] |
HCK proto-oncogene, Src family tyrosine kinase in Human [GtoPdb: 2032] [UniProtKB: P08631] | ||||||||
GtoPdb | - | - | 8.55 | pIC50 | 2.8 | nM | IC50 | J Med Chem (2016) 59: 4697-710 [PMID:27115835] |
LCK proto-oncogene, Src family tyrosine kinase in Human [GtoPdb: 2053] [UniProtKB: P06239] | ||||||||
GtoPdb | - | - | 9.3 | pIC50 | <0.5 | nM | IC50 | J Med Chem (2016) 59: 4697-710 [PMID:27115835] |
LYN proto-oncogene, Src family tyrosine kinase in Human [GtoPdb: 2060] [UniProtKB: P07948] | ||||||||
GtoPdb | - | - | 9.1 | pIC50 | 0.8 | nM | IC50 | J Med Chem (2016) 59: 4697-710 [PMID:27115835] |
SRC proto-oncogene, non-receptor tyrosine kinase in Human [GtoPdb: 2206] [UniProtKB: P12931] | ||||||||
GtoPdb | - | - | 9.3 | pIC50 | <0.5 | nM | IC50 | J Med Chem (2016) 59: 4697-710 [PMID:27115835] |
YES proto-oncogene 1, Src family tyrosine kinase in Human [GtoPdb: 2284] [UniProtKB: P07947] | ||||||||
GtoPdb | - | - | 9.3 | pIC50 | <0.5 | nM | IC50 | J Med Chem (2016) 59: 4697-710 [PMID:27115835] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.