probe 1.1 [PMID: 24187130] [Ligand Id: 9191] activity data from GtoPdb

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  • κ receptor in Human [GtoPdb: 318] [UniProtKB: P41145]
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DB Assay description Assay Type Standard value Standard parameter Original value Original units Original parameter Reference
κ receptor in Human [GtoPdb: 318] [UniProtKB: P41145]
GtoPdb - - 9.6 pKi 0.25 nM Ki J. Biol. Chem. (2013) 288: 36703-16 [PMID:24187130]
GtoPdb Measuring βarrestin2 recruitment - 5.38 pEC50 4129 nM EC50 J. Biol. Chem. (2013) 288: 36703-16 [PMID:24187130]
GtoPdb Measuring [35S]GTPγS binding - 7.51 pEC50 31 nM EC50 J. Biol. Chem. (2013) 288: 36703-16 [PMID:24187130]

Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.