astressin [Ligand Id: 925] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| CRF1 receptor in Human [GtoPdb: 212] [UniProtKB: P34998] | ||||||||
| GtoPdb | - | - | 8.8 | pKd | - | - | - |
Eur J Biochem (1998) 258: 78-84 [PMID:9851694]; J Pharmacol Exp Ther (2001) 296: 113-20 [PMID:11123370]; J Pharmacol Exp Ther (1999) 288: 729-34 [PMID:9918582] |
| GtoPdb | - | - | 8.7 | pKi | 2 | nM | Ki | Front Neuroendocrinol (2014) 35: 161-70 [PMID:24269930] |
| GtoPdb | - | - | 9.14 | pIC50 | 0.72 | nM | IC50 | J Med Chem (2002) 45: 4737-47 [PMID:12361401] |
| CRF2 receptor in Human [GtoPdb: 213] [UniProtKB: Q13324] | ||||||||
| GtoPdb | - | - | 8.9 | pKd | - | - | - | J Pharmacol Exp Ther (2001) 296: 113-20 [PMID:11123370] |
| GtoPdb | - | - | 9.21 | pIC50 | 0.62 | nM | IC50 | J Med Chem (2002) 45: 4737-47 [PMID:12361401] |
| CRF2 receptor in Mouse [GtoPdb: 213] [UniProtKB: Q60748] | ||||||||
| GtoPdb | - | - | 9 | pKd | - | - | - | J Pharmacol Exp Ther (1999) 288: 729-34 [PMID:9918582] |
| CRF2 receptor in Rat [GtoPdb: 213] [UniProtKB: P47866] | ||||||||
| GtoPdb | - | - | 8.8 | pKd | - | - | - | J Pharmacol Exp Ther (1999) 288: 729-34 [PMID:9918582] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
