setmelanotide [Ligand Id: 9272] activity data from GtoPdb
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| DB | Assay description | Assay Type | Standard value | Standard parameter | Original value | Original units | Original parameter | Reference |
|---|---|---|---|---|---|---|---|---|
| MC1 receptor in Human [GtoPdb: 282] [UniProtKB: Q01726] | ||||||||
| GtoPdb | - | - | 8.41 | pKi | 3.9 | nM | Ki | Peptides (2009) 30: 1892-900 [PMID:19646498] |
| MC3 receptor in Human [GtoPdb: 284] [UniProtKB: P41968] | ||||||||
| GtoPdb | - | - | 8 | pKi | 10 | nM | Ki | Peptides (2009) 30: 1892-900 [PMID:19646498] |
| MC4 receptor in Human [GtoPdb: 285] [UniProtKB: P32245] | ||||||||
| GtoPdb | - | - | 8.68 | pKi | 2.1 | nM | Ki |
Peptides (2009) 30: 1892-900 [PMID:19646498]; Lancet Diabetes Endocrinol (2020) 8: 960-970 [PMID:33137293] |
| MC4 receptor in Rat [GtoPdb: 285] [UniProtKB: P70596] | ||||||||
| GtoPdb | - | - | 8.57 | pKi | 2.7 | nM | Ki | Peptides (2009) 30: 1892-900 [PMID:19646498] |
| MC5 receptor in Human [GtoPdb: 286] [UniProtKB: P33032] | ||||||||
| GtoPdb | - | - | 6.37 | pKi | 430 | nM | Ki | Peptides (2009) 30: 1892-900 [PMID:19646498] |
Our curators have not yet identified this ligand in ChEMBL, but you may find additional data by searching on the ChEMBL site using the ligand's name or structure.
